Glutaminyl Cyclase, Diseases, and Development of Glutaminyl
Por um escritor misterioso
Last updated 01 agosto 2024
![Glutaminyl Cyclase, Diseases, and Development of Glutaminyl](https://ars.els-cdn.com/content/image/1-s2.0-S0968089623003905-ga1.jpg)
Discovery of potential scaffolds for glutaminyl cyclase inhibitors: virtual screening, synthesis, and evaluation - ScienceDirect
![Glutaminyl Cyclase, Diseases, and Development of Glutaminyl](https://pubs.acs.org/cms/10.1021/acs.jmedchem.1c00325/asset/images/medium/jm1c00325_0003.gif)
Glutaminyl Cyclase, Diseases, and Development of Glutaminyl Cyclase Inhibitors
![Glutaminyl Cyclase, Diseases, and Development of Glutaminyl](https://www.mdpi.com/molecules/molecules-23-00924/article_deploy/html/images/molecules-23-00924-g001.png)
Molecules, Free Full-Text
Full article: Hypothesis: glutaminyl cyclase inhibitors decrease risks of Alzheimer's disease and related dementias
is a glutaminyl cyclase inhibitor with an IC50 of 0.5 μM.Glutaminyl Cyclase Inhibitor 1 is compound 23[1].[1]. Li M, et al. Synthesis and
![Glutaminyl Cyclase, Diseases, and Development of Glutaminyl](https://www.glpbio.com/media/struct/GC3/GC30892.png)
Glutaminyl Cyclase Inhibitor 1
![Glutaminyl Cyclase, Diseases, and Development of Glutaminyl](https://static.hindawi.com/articles/bmri/volume-2022/4154697/figures/4154697.fig.003c.jpg)
Upregulation of Glutaminyl Cyclase Contributes to ERS-Induced Apoptosis in PC12 Cells
![Glutaminyl Cyclase, Diseases, and Development of Glutaminyl](https://media.springernature.com/lw685/springer-static/image/art%3A10.1007%2Fs00401-021-02349-5/MediaObjects/401_2021_2349_Fig4_HTML.png)
A glutaminyl cyclase-catalyzed α-synuclein modification identified in human synucleinopathies
![Glutaminyl Cyclase, Diseases, and Development of Glutaminyl](https://media.springernature.com/m685/springer-static/image/art%3A10.1038%2Fs41380-021-01409-2/MediaObjects/41380_2021_1409_Fig1_HTML.png)
Pyroglutamate Aβ cascade as drug target in Alzheimer's disease
![Glutaminyl Cyclase, Diseases, and Development of Glutaminyl](https://www.frontiersin.org/files/Articles/1209863/fnagi-15-1209863-HTML/image_m/fnagi-15-1209863-t004.jpg)
Frontiers Development and evolution of human glutaminyl cyclase inhibitors (QCIs): an alternative promising approach for disease-modifying treatment of Alzheimer's disease
![Glutaminyl Cyclase, Diseases, and Development of Glutaminyl](https://pubs.acs.org/cms/10.1021/acs.jmedchem.1c00325/asset/images/large/jm1c00325_0004.jpeg)
Glutaminyl Cyclase, Diseases, and Development of Glutaminyl Cyclase Inhibitors
![Glutaminyl Cyclase, Diseases, and Development of Glutaminyl](https://www.researchgate.net/profile/Manfred-Windisch/publication/23300963/figure/fig4/AS:281183029088269@1444050666435/Glutaminyl-cyclase-expression-and-pE-A-in-Alzheimers-disease-prevention-of-pE-A_Q320.jpg)
Glutaminyl cyclase expression and pE-A in Alzheimer's disease
![Glutaminyl Cyclase, Diseases, and Development of Glutaminyl](https://www.future-science.com/cms/10.4155/fmc.2019.11.issue-24/asset/17b34429-0617-3442-a061-b34429a0617b/cover.jpg)
An overview of glutaminyl cyclase inhibitors for Alzheimer's disease
![Glutaminyl Cyclase, Diseases, and Development of Glutaminyl](https://jpet.aspetjournals.org/sites/default/files/highwire/jpet/362/1.cover-source.jpg)
Glutaminyl Cyclase Inhibitor PQ912 Improves Cognition in Mouse Models of Alzheimer's Disease—Studies on Relation to Effective Target Occupancy
![Glutaminyl Cyclase, Diseases, and Development of Glutaminyl](https://i1.rgstatic.net/publication/317422052_Glutaminyl_cyclase_activity_correlates_with_levels_of_Ab_peptides_and_mediators_of_angiogenesis_in_cerebrospinal_fluid_of_Alzheimer's_disease_patients/links/595f39ca0f7e9b8194b73d09/largepreview.png)
PDF) Glutaminyl cyclase activity correlates with levels of Aβ peptides and mediators of angiogenesis in cerebrospinal fluid of Alzheimer's disease patients
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